Peptide Active Data Details
Basic Peptide Information
DICL ID
DICL_Pep_00890
Ion Channel
Neuronal acetylcholine receptor subunit alpha-3/beta-2
Peptide Function
Blocker
Gene Name
CHRNA3/CHRNB2
Activity Data (nM)
IC50
9.7 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified
Sequence Information
Peptide Sequence
GCCSHPACSVNHPELC
Peptide UniProt Accession
UniParc
UPI0001874811
Peptide Synonyms/Alias
α-PeIA
Peptide Species
Conus pergrandis (Grand cone)
Peptide Name
Alpha-conotoxin PeIA
CAS Number
Not available
Experimental Conditions
pH
Not mention
Holding Potential (mV)
−70 mV
Temperature
Not mention
Test Method
Patch-clamping
Test Species
Xenopus laevis oocyte
Binding Information
Binding Site
Not specified
Binding Site Residue
Not specified
Ion Channel Information
Gene Abbreviation (ABB)
nAChRs
Ion Channel UniProt Accession
Source Organism
Rattus norvegicus (Rat)
References & Disease Information
Disease
Not specified
PubChem CID
Not available
URL
Not available
PMID
Patent
Not available